SCHEMBL3656307

SCHEMBL3656307

CC(C)(C)C(=O)Nc1ccc(C(=O)CN2C(=O)NC(Cc3ccccc3)(c3ccccc3)C2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.53
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.44
PKM P14618 1/20 0.44
USP2 O75604 1/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3662076 0.87 KMT2A (0.55) HDAC6KMT2AMEN1POLBPKM
SCHEMBL3662282 0.86 HDAC6 (0.53) HDAC6KMT2AMEN1POLBPKM
SCHEMBL3662021 0.84 HDAC6 (0.51) HDAC6KMT2AMEN1POLBPKM
SCHEMBL3659938 0.79 KMT2A (0.61) KMT2AMEN1POLBPKMUSP2
SCHEMBL3660710 0.78 KMT2A (0.66) KMT2AMEN1POLBPKMUSP2
SCHEMBL3663347 0.77 KMT2A (0.58) HDAC6KMT2AMEN1LMNAPOLB
SCHEMBL4121157 0.76 KMT2A (0.55) HDAC6KMT2AMEN1LMNAUSP2
SCHEMBL3664165 0.75 KMT2A (0.52) HDAC6KMT2AMEN1LMNAPOLB
SCHEMBL3660498 0.74 KMT2A (0.61) KMT2AMEN1POLBPKMUSP2
SCHEMBL3796712 0.74 HDAC6 (0.46) HDAC6KMT2AMEN1POLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101827840-A Imidazolidine-2,4-dione (hydantoin) derivatives useful as npy y2 receptor modulators NOVARTIS AG 2010-09-08 CN claimed
EP-2212314-A1 IMIDAZOLIDINE-2,4-DIONE (HYDANTOIN) DERIVATIVES USEFUL AS NPY Y2 RECEPTOR MODULATORS Novartis AG (CH) 2010-08-04 EP claimed
WO-2009050200-A1 IMIDAZOLIDINE-2,4-DIONE (HYDANTOIN) DERIVATIVES USEFUL AS NPY Y2 RECEPTOR MODULATORS NOVARTIS AG (CH) 2009-04-23 WO claimed
US-20090099243-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-04-16 US claimed
CN-101827840-A Imidazolidine-2,4-dione (hydantoin) derivatives useful as npy y2 receptor modulators NOVARTIS AG 2010-09-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099243-A1 ORGANIC COMPOUNDS SLCO4C1, SLCO1B1, SLCO1B3 HDAC6 715/4885KMT2A 2020/4885MEN1 155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.