SCHEMBL365665

SCHEMBL365665

COCCNC(=O)c1ccc2c(C(=O)O)c3ccccn3c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.50
ACSS2 Q9NR19 1/20 0.46
KDM4E B2RXH2 4/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
MAPT P10636 1/20 0.45
DGAT2 Q96PD7 1/20 0.44
PPARG P37231 1/20 0.44
ALDH1A1 P00352 4/20 0.43
HSD17B10 Q99714 3/20 0.43
HTT P42858 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
TP53 P04637 3/20 0.43
ABL1 P00519 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
RIN1 Q13671 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364295 0.91 HPGD (0.47) HPGDACSS2KDM4ENPC1RAB9A
Potassium Ion SCHEMBL366533 0.89 HPGD (0.45) HPGDACSS2KDM4ENPC1RAB9A
SCHEMBL365908 0.87 KDM4E (0.45) HPGDACSS2KDM4ENPC1RAB9A
SCHEMBL31060260 0.87 KDM4E (0.45) HPGDACSS2KDM4ENPC1RAB9A
SCHEMBL366535 0.86 EGFR (0.48) HPGDACSS2KDM4EMAPTALDH1A1
SCHEMBL364233 0.84 KDM4E (0.44) HPGDACSS2KDM4ENPC1RAB9A
SCHEMBL365749 0.82 KDM4E (0.45) HPGDACSS2KDM4ENPC1RAB9A
SCHEMBL366370 0.82 EGFR (0.43) ACSS2KDM4EMAPTALDH1A1MEN1
SCHEMBL365666 0.82 HPGD (0.52) HPGDKDM4ERAB9APPARGALDH1A1
SCHEMBL361356 0.80 EGFR (0.47) HPGDACSS2KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed