SCHEMBL365666

SCHEMBL365666

COCCNC(=O)c1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.52
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 4/20 0.50
HSD17B10 Q99714 2/20 0.50
TP53 P04637 1/20 0.50
GLA P06280 1/20 0.50
GAA P10253 1/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
MAPK1 P28482 1/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
ABL1 P00519 1/20 0.44
CYP3A4 P08684 1/20 0.44
RIN1 Q13671 1/20 0.44
BRD4 O60885 1/20 0.43
KMT2A Q03164 1/20 0.43
PTGER4 P35408 1/20 0.43
PPARG P37231 1/20 0.43
ADORA2A P29274 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364296 0.91 ALDH1A1 (0.49) HPGDKDM4EALDH1A1HSD17B10TP53
Potassium Ion SCHEMBL366534 0.89 ALDH1A1 (0.47) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL365909 0.87 LMNA (0.45) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL366536 0.85 EGFR (0.53) HPGDKDM4EALDH1A1HSD17B10CYP1A2
SCHEMBL364234 0.83 ALDH1A1 (0.45) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL365665 0.82 HPGD (0.50) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL365750 0.81 POLB (0.46) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL366371 0.81 EGFR (0.45) HPGDKDM4EALDH1A1BRD4EGFR
SCHEMBL361357 0.79 EGFR (0.51) HPGDKDM4EALDH1A1HSD17B10TP53
SCHEMBL365935 0.78 KDM4E (0.47) HPGDKDM4EALDH1A1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed