SCHEMBL365778

SCHEMBL365778

CSc1ccc2c(C(=O)O)c3ccccn3c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.42
IDO1 P14902 3/20 0.42
DHODH Q02127 1/20 0.41
PTGS2 P35354 1/20 0.41
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
MEN1 O00255 4/20 0.40
MAPT P10636 4/20 0.40
KMT2A Q03164 4/20 0.40
SAE1 Q9UBE0 2/20 0.40
UBA2 Q9UBT2 2/20 0.40
APAF1 O14727 1/20 0.40
G6PD P11413 1/20 0.40
PABPC1 P11940 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
MCL1 Q07820 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
FNTA P49354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367704 0.87 EGFR (0.43) EGFRPTGS2ALDH1A1KDM4EMEN1
SCHEMBL365369 0.85 MAPT (0.47) EGFRIDO1ALDH1A1KDM4EMEN1
SCHEMBL365934 0.81 KDM4E (0.45) EGFRIDO1PTGS2ALDH1A1KDM4E
SCHEMBL366887 0.81 KDM4E (0.56) EGFRIDO1PTGS2ALDH1A1KDM4E
SCHEMBL366875 0.80 EGFR (0.42) EGFRIDO1PTGS2ALDH1A1KDM4E
SCHEMBL371112 0.80 IDO1 (0.51) EGFRIDO1PTGS2ALDH1A1KDM4E
SCHEMBL365013 0.79 KDM4E (0.58) EGFRALDH1A1KDM4EMEN1MAPT
SCHEMBL366810 0.78 PTGS2 (0.45) EGFRIDO1PTGS2ALDH1A1KDM4E
SCHEMBL365779 0.78 EGFR (0.43) EGFRDHODHALDH1A1KDM4EMEN1
SCHEMBL367746 0.78 EGFR (0.43) EGFRIDO1PTGS2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed