SCHEMBL365779

SCHEMBL365779

CSc1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
AGTR1 P30556 7/20 0.40
SRC P12931 5/20 0.39
DHODH Q02127 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
FGFR1 P11362 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367705 0.87 EGFR (0.48) EGFRKDM4EALDH1A1POLBAGTR1
SCHEMBL365370 0.85 NPC1 (0.47) EGFRKDM4EALDH1A1SRCMEN1
SCHEMBL366888 0.78 EGFR (0.44) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL365935 0.78 KDM4E (0.47) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL365778 0.78 EGFR (0.42) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL366876 0.78 EGFR (0.44) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL367114 0.77 ALDH1A1 (0.49) EGFRALDH1A1POLBHPGDSRC
SCHEMBL365014 0.77 KDM4E (0.48) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL367747 0.75 AGTR1 (0.48) EGFRKDM4EALDH1A1POLBHPGD
SCHEMBL366811 0.75 EGFR (0.44) EGFRKDM4EALDH1A1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed