SCHEMBL3657985

SCHEMBL3657985

COc1cccc(-c2cc(C(=O)O)cc(-c3nnn[nH]3)c2)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 2/20 0.49
ORAI1 Q96D31 2/20 0.49
ADORA3 P0DMS8 2/20 0.44
ADORA2A P29274 2/20 0.44
ADORA2B P29275 2/20 0.44
FFAR4 Q5NUL3 1/20 0.43
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
CTSA P10619 1/20 0.38
ABCB1 P08183 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
USP2 O75604 1/20 0.37
TPMT P51580 1/20 0.36
HAO1 Q9UJM8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655321 0.90 EGLN1 (0.43) ADORA3KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL3654728 0.82 CTSA (0.43) FFAR4CTSANPC1MAPTRAB9A
SCHEMBL3653036 0.81 STIM1 (0.45) STIM1ORAI1ADORA3KDM4EALDH1A1
SCHEMBL3649605 0.81 ALPL (0.51) KDM4EALDH1A1CTSASMN1; SMN2HAO1
SCHEMBL3655711 0.80 PTGER1 (0.44) ALDH1A1HPGDCTSATP53MAPT
SCHEMBL3652824 0.80 ALDH1A1 (0.44) KDM4EHSD17B10ALDH1A1HPGDCTSA
SCHEMBL3655146 0.80 CBFB (0.36) KDM4EALDH1A1TPMTHAO1MEN1
SCHEMBL3655959 0.80 ADORA3 (0.42) ADORA3KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL3652857 0.79 NR1H4 (0.43) NPC1RAB9ASMN1; SMN2ALPL
SCHEMBL3655999 0.79 ALPL (0.46) KDM4EHPGDNPC1TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP claimed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO claimed
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO disclosed