SCHEMBL3658151

SCHEMBL3658151

NCC(=O)OC(=O)[C@@H](N)Cc1c[nH]c2ccc(O)cc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.67
NPSR1 Q6W5P4 5/20 0.67
HTR1A P08908 4/20 0.67
HTR2A P28223 4/20 0.67
HTR2B P41595 4/20 0.67
TSHR P16473 4/20 0.67
BLM P54132 4/20 0.67
MAPT P10636 4/20 0.67
NFKB1 P19838 3/20 0.67
CYP3A4 P08684 3/20 0.67
LMNA P02545 3/20 0.67
PMP22 Q01453 3/20 0.67
ALDH1A1 P00352 3/20 0.67
KMT2A Q03164 3/20 0.67
KDM4E B2RXH2 3/20 0.67
HTR7 P34969 2/20 0.67
ADORA3 P0DMS8 1/20 0.67
ALOX15 P16050 1/20 0.67
SLC6A4 P31645 1/20 0.67
MTOR P42345 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19357216 0.91 HTR2C (0.76) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL2721523 0.86 BLM (0.67) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL30472798 0.85 NPSR1 (0.64) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL20657043 0.85 NPSR1 (0.64) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL13282480 0.84 HTR2C (0.69) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL471920 0.84 NPSR1 (0.72) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL6775810 0.84 NPSR1 (0.72) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL424584 0.84 MAPT (0.65) HTR2CHTR1AHTR2AHTR2BTSHR
SCHEMBL816987 0.83 NPSR1 (0.70) HTR2CNPSR1HTR1AHTR2AHTR2B
SCHEMBL10407437 0.83 NPSR1 (0.70) HTR2CNPSR1HTR1AHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200997-A1 SYNTHESIS OF DEUTERATED CATECHOLS AND BENZOÝD¨Ý1,3¨DIOXOLES AND DERIVATIVES THEREOF Concert Pharmaceuticals Inc. (US) 2010-06-30 EP disclosed
WO-2009035652-A1 SYNTHESIS OF DEUTERATED CATECHOLS AND BENZO[D][1,3] DIOXOLES AND DERIVATIVES THEREOF CONCERT PHARMACEUTICALS, INC. (US) 2009-03-19 WO disclosed