SCHEMBL3658282

SCHEMBL3658282

COc1cc(C(N)=O)ccc1-c1ccnc(N)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.54
MKNK2 Q9HBH9 1/20 0.54
JAK2 O60674 1/20 0.49
MAPK1 P28482 1/20 0.48
CCNT1 O60563 3/20 0.47
CDK9 P50750 3/20 0.47
CDK2 P24941 2/20 0.47
CDC7 O00311 2/20 0.47
CSNK2A2 P19784 1/20 0.47
CCNE1 P24864 1/20 0.47
CSNK1A1 P48729 1/20 0.47
CSNK1D P48730 1/20 0.47
CSNK2B P67870 1/20 0.47
CSNK2A1 P68400 1/20 0.47
DBF4 Q9UBU7 1/20 0.47
CDK5 Q00535 2/20 0.47
CDK5R1 Q15078 2/20 0.47
CCNA2 P20248 1/20 0.47
CCNA1 P78396 1/20 0.47
GSK3B P49841 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658285 0.80 CCNT1 (0.53) JAK2CCNT1CDK9CDK2CDK5
SCHEMBL30507464 0.79 GSK3B (0.60) MAPK1CCNT1CDK9CDK2CDC7
SCHEMBL28512792 0.79 GSK3B (0.60) MAPK1CCNT1CDK9CDK2CDC7
SCHEMBL28497712 0.79 CDK2 (0.52) CCNT1CDK9CDK2CDC7CCNE1
SCHEMBL30507501 0.79 CDK2 (0.52) CCNT1CDK9CDK2CDC7CCNE1
SCHEMBL15939816 0.78 CHRNA7 (0.55) CCNT1CDK9CDK2CDK5CDK5R1
SCHEMBL30507254 0.78 CHRNA7 (0.55) CCNT1CDK9CDK2CDK5CDK5R1
SCHEMBL3362587 0.74 HSP90AA1 (0.60) CCNT1CDK9CDK2CDK5CDK5R1
SCHEMBL30507329 0.74 HSP90AA1 (0.60) CCNT1CDK9CDK2CDK5CDK5R1
SCHEMBL8842473 0.74 PRSS1 (0.48) MKNK1MKNK2CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed