SCHEMBL3659396

SCHEMBL3659396

N#Cc1ccc(-c2ccc[c]c2C(N)=O)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 15/20 0.49
CYP11B1 P15538 14/20 0.42
SLC22A12 Q96S37 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
STAT3 P40763 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39
TUBA1A Q71U36 1/20 0.39
TUBA1C Q9BQE3 1/20 0.39
TUBB6 Q9BUF5 1/20 0.39
TUBB2B Q9BVA1 1/20 0.39
TUBB1 Q9H4B7 1/20 0.39
KDM1A O60341 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660537 0.90 CNR2 (0.43) CYP11B2
SCHEMBL4630355 0.78 IRAK4 (0.41) CYP11B2CYP11B1
SCHEMBL3097233 0.77 IKBKB (0.46) SLC22A12
SCHEMBL3653879 0.76 CDC7 (0.40)
SCHEMBL3462201 0.76 GRM2 (0.41)
SCHEMBL3663745 0.75 SLC9A1 (0.42)
SCHEMBL27710717 0.71 CYP11B2 (0.54) CYP11B2CYP11B1
SCHEMBL2636302 0.71 BCAT2 (0.53)
SCHEMBL3304437 0.71 CYP11B1 (0.72) CYP11B2CYP11B1TUBB4ATUBBTUBA3C
SCHEMBL4911450 0.71 PARP1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8642788-B2 Activators of executioner procaspases 3, 6 and 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-02-04 US disclosed
EP-2237784-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 The Regents of the University of California (US) 2010-10-13 EP disclosed
WO-2009089508-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-07-16 WO disclosed