SCHEMBL3660736

SCHEMBL3660736

CC(C)CC1c2cccc(C(=N)NO)c2CN1C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.35
ABCB1 P08183 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
MTNR1B P49286 1/20 0.32
ACE P12821 1/20 0.32
HHAT Q5VTY9 2/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2126330 0.89 ABCB1 (0.39) HDAC6ABCB1ABCG2MTNR1BACE
SCHEMBL2122271 0.79 ABCB1 (0.37) HDAC6ABCB1ABCG2MTNR1BHHAT
SCHEMBL3660735 0.78
SCHEMBL3664397 0.76 NOTUM (0.36) ABCB1ABCG2MTNR1BACEKDM4E
SCHEMBL2122064 0.71 ABCB1 (0.43) ABCB1ABCG2MTNR1BACEHHAT
SCHEMBL3657289 0.70 MTNR1B (0.37) HDAC6MTNR1B
SCHEMBL2126327 0.69 PKM (0.32) KDM4E
SCHEMBL2121421 0.69 KIF11 (0.38) MTNR1BACE
SCHEMBL2121308 0.65 ESR1 (0.34) ABCB1ABCG2
SCHEMBL2122590 0.64 ESR1 (0.47) ABCB1ABCG2MTNR1BHHATKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222670-A1 OXADIAZOLE DERIVATIVES FOR USE AS S1P1 AGONISTS IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS Glaxo Group Limited (GB) 2010-09-01 EP disclosed
WO-2009080729-A1 OXADIAZOLE DERIVATIVES FOR USE AS S1P1 AGONISTS IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed