SCHEMBL3660901

SCHEMBL3660901

CC(C)(C)OC(=O)NCC(C#N)c1ccc(-c2cccc(C#N)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.48
CTSK P43235 4/20 0.48
CTSB P07858 2/20 0.48
MCHR1 Q99705 12/20 0.45
ADAMTS4 O75173 1/20 0.41
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
CTSL P07711 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5170834 0.80 CTSS (0.61) CTSSCTSKCTSBCTSL
SCHEMBL2074657 0.79 CTSC (0.57) CTSSCTSKCTSBMMP12MMP13
SCHEMBL2074655 0.79 CTSC (0.57) CTSSCTSKCTSBMMP12MMP13
SCHEMBL3654576 0.78 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL3651290 0.78 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL6028072 0.78 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL3661255 0.76 CTSC (0.47) CTSKMCHR1
SCHEMBL30771381 0.76 CTSS (0.47) CTSSCTSKCTSBCTSL
SCHEMBL3715972 0.75 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL31724229 0.75 CTSS (0.44) CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231597-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2010-09-29 EP disclosed
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed