SCHEMBL3660967

SCHEMBL3660967

C=C1CN(Cc2ccccc2)Cc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
SIGMAR1 Q99720 5/20 0.47
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
MC4R P32245 1/20 0.44
ACHE P22303 2/20 0.43
CYP1A2 P05177 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6672942 0.81 SIGMAR1 (0.62) SIGMAR1MC4RACHECYP1A2HTR2C
SCHEMBL4000995 0.79 SIGMAR1 (0.54) MAPTTDP1SIGMAR1MC4RACHE
Hydrochloric Acid SCHEMBL16713355 0.79 SIGMAR1 (0.60) SIGMAR1MC4RACHECYP1A2HTR2C
SCHEMBL30978695 0.75 SIGMAR1 (0.60) TDP1SIGMAR1MC4RACHE
SCHEMBL30073105 0.75 SIGMAR1 (0.60) SIGMAR1MC4RCYP1A2MEN1KMT2A
SCHEMBL20060315 0.74 NR3C1 (0.45) MAPTTDP1SIGMAR1ADRA1DADRA1A
SCHEMBL8450698 0.74 SIGMAR1 (0.58) TDP1SIGMAR1MC4RACHECYP1A2
SCHEMBL12773114 0.72 ADRA1D (0.42) MAPTTDP1ADRA1DADRA1AADRA1B
SCHEMBL3240403 0.71 MEN1 (0.46) SIGMAR1MC4RACHEMEN1KMT2A
SCHEMBL17618300 0.70 SIGMAR1 (0.50) SIGMAR1ADRA1DADRA1AADRA1BMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215064-A1 COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY Schering Corporation (US) 2010-08-11 EP disclosed
WO-2009061596-A1 COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY SCHERING CORPORATION (US) 2009-05-14 WO disclosed