SCHEMBL3661830

SCHEMBL3661830

COc1ccc(C(Cc2ccnc(-c3ccc(C(=O)O)cc3)c2)C(O)C(F)(F)F)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.43
MRGPRX4 Q96LA9 1/20 0.39
HDAC1 Q13547 4/20 0.37
KDM1A O60341 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC5 Q9UQL6 2/20 0.37
CHEK1 O14757 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTPN1 P18031 2/20 0.37
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660214 0.92 MRGPRX4 (0.44) MRGPRX4KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL3652326 0.90 CDC7 (0.39) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL3654236 0.81 LOXL2 (0.37) LOXL2MRGPRX4HDAC1KDM1AHDAC6
SCHEMBL3651279 0.79 KMO (0.39) LOXL2MRGPRX4RORCKMOKDM5A
SCHEMBL3657608 0.77 EIF4E (0.36) LOXL2KMOKDM4C
SCHEMBL3659044 0.77 MRGPRX4 (0.38) MRGPRX4
SCHEMBL3659842 0.76 KMO (0.36) LOXL2MRGPRX4KMO
SCHEMBL837203 0.76 CHEK1 (0.39) LOXL2MRGPRX4HDAC1KDM1AHDAC6
SCHEMBL3658104 0.73 MRGPRX4 (0.42) MRGPRX4KDM4EALDH1A1NPC1RAB9A
SCHEMBL3653818 0.73 CDC7 (0.38) MRGPRX4KDM4EALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed