SCHEMBL3661903

SCHEMBL3661903

COC(=O)NC1CC=C(c2c[nH]c3cccnc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.44
HTR1E P28566 2/20 0.42
HTR1A P08908 1/20 0.42
ROCK2 O75116 1/20 0.41
CDK7 P50613 1/20 0.40
CDK9 P50750 1/20 0.40
JAK1 P23458 2/20 0.37
SLC6A4 P31645 2/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
NOS3 P29474 2/20 0.36
NOS1 P29475 2/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951141 0.90 HTR1D (0.41) HTR1DHTR1EHTR1AROCK2CDK7
SCHEMBL3211442 0.88 HTR1D (0.46) HTR1DHTR1EHTR1AROCK2CDK7
SCHEMBL3214716 0.83 NOS3 (0.46) HTR1DHTR1EHTR1ACDK7CDK9
SCHEMBL3217678 0.82 CDK7 (0.45) HTR1DHTR1EHTR1AROCK2CDK7
SCHEMBL3214861 0.79 JAK3 (0.39) HTR1DHTR1EHTR1AROCK2CDK7
SCHEMBL3653965 0.78 HTR1D (0.41) HTR1DHTR1EHTR1ACDK7CDK9
SCHEMBL3216008 0.77 JAK2 (0.44) HTR1DHTR1EHTR1ACDK7CDK9
SCHEMBL3348186 0.75 ROCK2 (0.46) ROCK2CDK7CDK9JAK1KDR
SCHEMBL3227327 0.74 SLC6A4 (0.66) HTR1DCDK7CDK9SLC6A4KDR
SCHEMBL3211296 0.73 SLC6A4 (0.45) HTR1DHTR1EHTR1ASLC6A4NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010024980-A1 4'-AMINO CYCLIC COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY MEMORY PHARMACEUTICALS CORPORATION (US) 2010-03-04 WO disclosed