SCHEMBL3661937

SCHEMBL3661937

O=C(O)c1cc(Br)cc(C(O)(C(F)(F)F)C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.46
POLB P06746 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
P2RY14 Q15391 1/20 0.39
TTR P02766 1/20 0.38
SRD5A2 P31213 2/20 0.36
NR1H3 Q13133 2/20 0.36
NR1H2 P55055 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
MLYCD O95822 4/20 0.35
RORC P51449 1/20 0.35
CES2 O00748 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNJ11 Q14654 1/20 0.34
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14593293 0.87 CES2 (0.45) SRD5A2NR1H3NR1H2RXRARXRB
SCHEMBL1333906 0.87 LCK (0.43) SRD5A2NR1H3NR1H2RXRARXRB
Hydrochloric Acid SCHEMBL15948160 0.85 LCK (0.42) SRD5A2NR1H3NR1H2RXRARXRB
SCHEMBL494019 0.83 NOTUM (0.64) NOTUMPOLBHCAR2P2RY14TTR
SCHEMBL1332001 0.80 AR (0.41) NOTUMNR1H3NR1H2MLYCDRORC
SCHEMBL23411745 0.80 NOTUM (0.51) NOTUMPOLBHCAR2P2RY14TTR
SCHEMBL29728800 0.80 NOTUM (0.51) NOTUMPOLBHCAR2P2RY14TTR
SCHEMBL23411618 0.80 NOTUM (0.51) NOTUMPOLBHCAR2P2RY14TTR
SCHEMBL29728806 0.80 NOTUM (0.51) NOTUMPOLBHCAR2P2RY14TTR
SCHEMBL3072277 0.78 NOTUM (0.45) NOTUMPOLBHCAR2P2RY14TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215049-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN Merck Sharp & Dohme Corp. (US) 2010-08-11 EP disclosed
WO-2009058298-A1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK & CO., INC. (US) 2009-05-07 WO disclosed