SCHEMBL3662419

SCHEMBL3662419

COc1ccc(C2=CC=CC(C)(N)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
ESR2 Q92731 1/20 0.35
DYRK1A Q13627 1/20 0.35
MAPK1 P28482 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
APP P05067 2/20 0.34
MAOB P27338 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOA P21397 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990190 0.76
SCHEMBL7609289 0.76 SLC6A3 (0.40) CA1CA2ESR2ALDH1A1KMT2A
SCHEMBL5135826 0.67 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL28526225 0.66 NPC1 (0.32) ALDH1A1
SCHEMBL28447735 0.65 PTGS2 (0.36) PTGS1PTGS2MEN1KMT2ASMN1; SMN2
SCHEMBL28239119 0.64 CA1 (0.55) CA12CA1CA2CA7CA9
SCHEMBL29170920 0.63 NPC1 (0.42) MAPK1TDP1MAOBALDH1A1MAOA
SCHEMBL28567153 0.63 NPC1 (0.36) ALDH1A1
SCHEMBL8884493 0.63 CA1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL22288164 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2237784-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 The Regents of the University of California (US) 2010-10-13 EP disclosed
WO-2009089508-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-07-16 WO disclosed