SCHEMBL3662545

SCHEMBL3662545

COc1ccc2cnn(N)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.57
HTR2C P28335 2/20 0.57
HTR2B P41595 1/20 0.57
CA2 P00918 1/20 0.43
CYP1A2 P05177 3/20 0.42
CYP2A6 P11509 1/20 0.42
NCF1 P14598 1/20 0.42
PIM3 Q86V86 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ROCK1 Q13464 1/20 0.41
EGFR P00533 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
POLB P06746 2/20 0.41
MAPK1 P28482 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13113212 0.80 HTR2A (0.59) HTR2AHTR2CHTR2BCA2CYP1A2
SCHEMBL28707949 0.76 HTR2A (0.67) HTR2AHTR2CHTR2BCYP1A2CYP2A6
SCHEMBL3656364 0.76 KMO (0.51) HTR2AHTR2CHTR2BCYP1A2CYP2A6
SCHEMBL6364886 0.73 HTR2C (1.00) HTR2AHTR2CHTR2B
SCHEMBL7006841 0.73 HTR2C (0.59) HTR2AHTR2CHTR2BCA2PIM3
SCHEMBL31079387 0.73 HTR2C (1.00) HTR2AHTR2CHTR2B
SCHEMBL4953169 0.73 CHEK1 (0.42) HTR2AHTR2CHTR2BPIM3MAPT
SCHEMBL30816402 0.72 HTR2A (0.62) HTR2AHTR2CHTR2BPIM3MAPT
SCHEMBL27165386 0.72 HTR2A (0.62) HTR2AHTR2CHTR2BPIM3MAPT
SCHEMBL17454422 0.72 KMO (0.51) HTR2AHTR2CHTR2BCYP2A6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227464-A1 DERIVATIVES OF 1-[(IMIDAZOLIDIN-2-YL)IMINO)]INDAZOLE Imperial Innovations Limited (GB) 2010-09-15 EP disclosed
WO-2009071906-A1 DERIVATIVES OF 1-[(IMIDAZOLIDIN-2-YL)IMINO)]INDAZOLE IMPERIAL INNOVATIONS LIMITED (GB) 2009-06-11 WO disclosed