SCHEMBL3663573

SCHEMBL3663573

COc1cccc2c1oc1ccc([N+](=O)[O-])cc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.52
RAB9A P51151 3/20 0.52
NPC1 O15118 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
ADORA3 P0DMS8 1/20 0.50
ADORA2A P29274 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPT P10636 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
HTT P42858 1/20 0.47
HNF4A P41235 2/20 0.46
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11385812 0.91 MAOA (0.63) MAOARAB9ANPC1KDM4EALDH1A1
SCHEMBL5738370 0.80 MAOA (0.48) MAOARAB9ANPC1KDM4EALDH1A1
SCHEMBL1750256 0.76 PTPN1 (0.46) RAB9ANPC1KDM4EALDH1A1LMNA
SCHEMBL1751525 0.75 ALDH1A1 (0.48) MAOARAB9ANPC1ALDH1A1LMNA
SCHEMBL2340821 0.75 MAPT (0.81) RAB9ANPC1KDM4EALDH1A1MEN1
SCHEMBL1750895 0.74 HTT (0.43) RAB9ANPC1ALDH1A1LMNAL3MBTL1
Hydrochloric Acid SCHEMBL4026672 0.74 ALDH1A1 (0.47) MAOARAB9ANPC1ALDH1A1LMNA
SCHEMBL1301907 0.74 MAOA (0.75) MAOARAB9ANPC1KDM4EALDH1A1
SCHEMBL11093874 0.74 HNF4A (0.60) MAOARAB9ANPC1KDM4EALDH1A1
SCHEMBL7233246 0.74 HTT (0.51) MAOARAB9AKDM4EALDH1A1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225205-A1 ESTER DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.p.A. (IT) 2010-09-08 EP disclosed
WO-2009077068-A9 ESTER DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMA SPA (IT) 2009-08-20 WO disclosed
WO-2009077068-A1 ESTER DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2009-06-25 WO disclosed