SCHEMBL3663718

SCHEMBL3663718

COc1cnc2nc(-c3cnc4c(c3)CCC(NC(=O)O)C4)c(=O)[nH]c2c1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
IKBKE Q14164 8/20 0.34
TBK1 Q9UHD2 8/20 0.34
MAPK1 P28482 1/20 0.33
GRIN1 Q05586 4/20 0.33
GRIN2B Q13224 4/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
ACHE P22303 2/20 0.33
AURKB Q96GD4 3/20 0.33
CDK2 P24941 1/20 0.32
HDAC8 Q9BY41 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3667973 0.76 HDAC1 (0.32) HDAC8
SCHEMBL3669837 0.76 AURKA (0.32) IKBKETBK1AURKBCDK2
SCHEMBL3019050 0.76 KCNH2 (0.46)
SCHEMBL3022635 0.73 MTNR1A (0.36) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL3020759 0.69 MTNR1A (0.38) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL3663681 0.69 PDE2A (0.37) MTNR1AMTNR1BMAPK1CA1CA2
SCHEMBL3016078 0.68 MTNR1A (0.35) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL3016071 0.68 MTNR1A (0.35) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL3008126 0.68 MTNR1A (0.34) MTNR1AMTNR1BMAPK1CA1CA2
SCHEMBL3009533 0.66 MTNR1A (0.36) MTNR1AMTNR1BMAPK1GRIN2BCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139898-A1 COMPOUNDS Glaxo Group Limited (GB) 2010-01-06 EP disclosed
WO-2008128961-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed