SCHEMBL3664792

SCHEMBL3664792

O=C(CSC1=NCCS1)c1ccc2[nH]c3nc(Cl)ccc3c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
MAPT P10636 7/20 0.56
SMN1; SMN2 Q16637 3/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
KMT2A Q03164 4/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 2/20 0.40
PKM P14618 3/20 0.38
LMNA P02545 6/20 0.38
TDP1 Q9NUW8 2/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL675381 0.84 MAPT (0.58) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL674811 0.81 ALDH1A1 (0.55) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL675108 0.80 CA1 (0.46) ALDH1A1MAPTRAB9ANPC1KMT2A
SCHEMBL13464069 0.79 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL675624 0.77 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL16241842 0.76 GCGR (0.63) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL3665386 0.76 MAPT (0.39) ALDH1A1MAPTRAB9AKMT2AHPGD
SCHEMBL675067 0.76 ALPL (0.58) ALDH1A1MAPTSMN1; SMN2RAB9ANPC1
SCHEMBL676048 0.76 GSK3B (0.41) ALDH1A1MAPTSMN1; SMN2RAB9AKMT2A
SCHEMBL3665281 0.76 KDM4E (0.39) ALDH1A1KMT2AHPGDMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed