SCHEMBL3665281

SCHEMBL3665281

CN(C)CCSCC(=O)c1ccc2[nH]c3nc(Cl)ccc3c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TLR9 Q9NR96 8/20 0.36
TLR8 Q9NR97 8/20 0.36
TLR7 Q9NYK1 8/20 0.36
JAK2 O60674 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
HRH3 Q9Y5N1 2/20 0.34
KMT2A Q03164 2/20 0.33
MAPK1 P28482 1/20 0.33
RAD52 P43351 1/20 0.33
TERT O14746 1/20 0.33
MEN1 O00255 1/20 0.32
GCGR P47871 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL678686 0.90 TERT (0.35) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL675224 0.85 ALDH1A1 (0.38) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL675928 0.83 KDM4E (0.39) KDM4EALDH1A1HPGDHSD17B10TLR9
Diethylamine SCHEMBL3664811 0.82 HDAC3 (0.35) KDM4EALDH1A1KMT2AMEN1GCGR
SCHEMBL3665277 0.82 MAPT (0.33) KDM4EALDH1A1HSD17B10TLR8TLR7
SCHEMBL678859 0.82 KDM4E (0.44) KDM4EALDH1A1HPGDHSD17B10TLR9
SCHEMBL3665283 0.81 KIF11 (0.35) ALDH1A1KMT2AMEN1GCGRHDAC3
SCHEMBL3668532 0.80 TLR9 (0.42) KDM4EALDH1A1HPGDHSD17B10TLR9
SCHEMBL3670189 0.80 PKM (0.40) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL3664810 0.78 MEN1 (0.33) KDM4EALDH1A1HPGDHSD17B10TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed