SCHEMBL3664922

SCHEMBL3664922

COc1ccc(N)c(Nc2ccc3c(c2)CCCC3C)n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.37
BACE2 Q9Y5Z0 3/20 0.37
EGFR P00533 5/20 0.34
LCK P06239 2/20 0.34
PIK3CA P42336 8/20 0.34
HRH2 P25021 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
PIK3CD O00329 5/20 0.32
PIK3CB P42338 5/20 0.32
PIK3CG P48736 5/20 0.32
PIM1 P11309 1/20 0.32
MTOR P42345 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664919 0.88 BACE1 (0.36) BACE1BACE2EGFRLCKPIK3CA
SCHEMBL3667380 0.78 MAPK8 (0.33) BACE1BACE2EGFRPIK3CA
SCHEMBL3025404 0.77 KDM4C (0.40)
SCHEMBL3667381 0.76 KDM4C (0.35) BACE1BACE2
SCHEMBL2947601 0.70 NR4A1 (0.56)
SCHEMBL15825116 0.69 BRD4 (0.38) HRH2HRH3DRD2DRD1
SCHEMBL30931435 0.69 BRD4 (0.38) HRH2HRH3DRD2DRD1
SCHEMBL6811822 0.69 ALDH1A1 (0.45) EGFRLCK
SCHEMBL12891719 0.68 DRD2 (0.40) HRH2HRH3DRD2DRD1
SCHEMBL2267169 0.68 NPY5R (0.44) BACE1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139898-A1 COMPOUNDS Glaxo Group Limited (GB) 2010-01-06 EP disclosed
WO-2008128961-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed