SCHEMBL3665479

SCHEMBL3665479

O=C(O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1CCCN(Cc1ccccc1)Cc1cccc(OCc2ccccc2)c1.O=C(O)N1CC[C@H](n2c(=O)[nH]c3ccccc32)C(CCCN(Cc2ccccc2)Cc2ccccn2)C1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.37
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
OPRM1 P35372 2/20 0.36
CHRM1 P11229 4/20 0.33
DRD2 P14416 1/20 0.33
KCNH2 Q12809 1/20 0.33
PARP1 P09874 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CALCRL Q16602 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789708 1.00 HSD11B1 (0.37) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1838920 0.87 HSD11B1 (0.46) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1834964 0.87 BCHE (0.40) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1834967 0.87 OPRM1 (0.46) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1835882 0.87 OPRM1 (0.46) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1832648 0.85 OPRK1 (0.43) BCHEACHEOPRM1CHRM1DRD2
SCHEMBL1832267 0.85 OPRK1 (0.43) BCHEACHEOPRM1CHRM1DRD2
SCHEMBL1832646 0.85 BCHE (0.38) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL3397207 0.83 OPRM1 (0.47) HSD11B1BCHEACHEOPRM1CHRM1
SCHEMBL1833774 0.82 OPRM1 (0.42) HSD11B1BCHEACHEOPRM1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2160098-A2 USE OF COMPOUNDS HAVING A MONOGALACTOSYLDIACYLGLYCEROL SYNTHASE INHIBITORY ACTIVITY AS HERBICIDE OR ALGAECIDE, HERBICIDE AND ALGAECIDE COMPOSITIONS Commissariat a L'Energie Atomique (FR) 2010-03-10 EP disclosed
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP disclosed
WO-2008146174-A2 USE OF COMPOUNDS HAVING A MONOGALACTOSYLDIACYLGLYCEROL SYNTHASE INHIBITORY ACTIVITY AS HERBICIDE OR ALGAECIDE, HERBICIDE AND ALGAECIDE COMPOSITIONS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO disclosed