SCHEMBL3666054

SCHEMBL3666054

COc1ccc(C=Cc2ccc3c(c2)c2c(C=Cc4ccc(OC)cc4)ccnc2n3S(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 2/20 0.46
ALK Q9UM73 2/20 0.45
HDAC3 O15379 3/20 0.42
HDAC4 P56524 3/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC7 Q8WUI4 3/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC10 Q969S8 3/20 0.42
HDAC11 Q96DB2 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
HDAC9 Q9UKV0 3/20 0.42
HDAC5 Q9UQL6 3/20 0.42
HTR6 P50406 5/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
TRPA1 O75762 1/20 0.39
ADORA1 P30542 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676946 0.92 ALK (0.56) SNCAALKHDAC3HDAC4HDAC1
SCHEMBL678782 0.92 ALK (0.56) SNCAALKHDAC3HDAC4HDAC1
SCHEMBL3671974 0.91 IP6K1 (0.41) ALKHDAC3HDAC4HDAC1HDAC7
SCHEMBL675268 0.89 HDAC3 (0.41) SNCAHDAC3HDAC4HDAC1HDAC7
SCHEMBL3725129 0.84 HTR6 (0.42) SNCAHDAC3HDAC4HDAC1HDAC7
SCHEMBL3725130 0.84 HTR6 (0.42) SNCAHDAC3HDAC4HDAC1HDAC7
SCHEMBL674878 0.83 NFE2L2 (0.39) ALKHTR6PTGDR2
SCHEMBL16241826 0.80 HTR6 (0.42) SNCAHDAC3HDAC4HDAC1HDAC7
SCHEMBL3665338 0.80 HTR6 (0.42) SNCAHDAC3HDAC4HDAC1HDAC7
SCHEMBL675868 0.80 HTR6 (0.42) SNCAHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed