SCHEMBL3669424

SCHEMBL3669424

COCCCCn1c(O)nc2ncc(Cl)cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.37
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
PTBP1 P26599 1/20 0.35
CHEK1 O14757 1/20 0.34
WEE1 P30291 1/20 0.34
HRH4 Q9H3N8 8/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HRH3 Q9Y5N1 2/20 0.33
HTR3A P46098 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
HPGD P15428 2/20 0.33
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ITK Q08881 1/20 0.33
MCHR1 Q99705 1/20 0.32
NR3C1 P04150 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3666329 0.85 TLR8 (0.37) GAACHEK1WEE1HRH4TP53
SCHEMBL3667095 0.84 PSEN1 (0.39) GAAHRH4SMN1; SMN2KMT2A
SCHEMBL3670195 0.84 KDM4E (0.40) LMNAGAACHEK1WEE1HRH4
SCHEMBL3673651 0.84 APOBEC3G (0.38) HRH4TP53MAPTHRH3HTR3A
SCHEMBL3671987 0.82 NUDT1 (0.45) CHEK1WEE1HRH4MAPTHRH3
SCHEMBL3668071 0.82 HPGD (0.38) LMNAHRH4HRH3HTR3AHPGD
SCHEMBL3675495 0.81 HRH4 (0.41) CHEK1WEE1HRH4HRH3HTR3A
SCHEMBL3675941 0.79 KMT2A (0.42) HRH4HRH3HTR3AHPGDHTT
SCHEMBL3669322 0.78 HSP90B1 (0.37) HRH4HRH3HTR3AHPGDHTT
SCHEMBL3672462 0.78 HRH4 (0.36) HRH4MAPTHRH3HTR3AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139478-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Cytokinetics, Incorporated (US) 2010-01-06 EP claimed
WO-2008121333-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-10-09 WO claimed
US-20080242695-A1 Certain Chemical Entities, Compositions, and Methods CYTOKINETICS, INC. 2008-10-02 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242695-A1 Certain Chemical Entities, Compositions, and Methods TNNC1, TNNI3, TNNT2 PLAU 2228/4885LMNA 391/4885GAA 939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.