SCHEMBL3669859

SCHEMBL3669859

O=S(=O)(c1ccccc1)n1c2ccc(-c3ccco3)cc2c2ccc(Cl)nc21

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 2/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
KAT6A Q92794 2/20 0.37
SRC P12931 2/20 0.36
CYP3A4 P08684 1/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NR4A2 P43354 1/20 0.35
PTGES O14684 1/20 0.35
LMNA P02545 1/20 0.35
RECQL P46063 1/20 0.35
CXCL8 P10145 1/20 0.34
NOD1 Q9Y239 1/20 0.34
ALK Q9UM73 1/20 0.34
CHEK1 O14757 2/20 0.34
DCTPP1 Q9H773 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676078 0.88 ALDH1A1 (0.40) ALDH1A1HPGDTSHRHSD17B10KAT6A
SCHEMBL3668236 0.86 HTR6 (0.46) SRCCXCL8NOD1
SCHEMBL3666385 0.82 SRC (0.38) ALDH1A1HPGDTSHRHSD17B10KAT6A
SCHEMBL675472 0.82 SRC (0.43) SRC
SCHEMBL3664606 0.81 ALDH1A1 (0.37) ALDH1A1HPGDTSHRHSD17B10KAT6A
SCHEMBL3721458 0.81 CNR2 (0.37) ALDH1A1HPGDTSHRHSD17B10KAT6A
SCHEMBL675245 0.79 HTR6 (0.45) ALDH1A1TSHRKAT6AMAPTCXCL8
SCHEMBL675280 0.79 HTR6 (0.44) SRCMAPTSMN1; SMN2LMNACXCL8
SCHEMBL676831 0.78 ALDH1A1 (0.38) ALDH1A1HPGDTSHRHSD17B10KAT6A
SCHEMBL676610 0.77 ALDH1A1 (0.45) ALDH1A1MAPTNOD1DCTPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed