SCHEMBL3721458

SCHEMBL3721458

CCCCCc1ccc2c3cc(-c4ccco4)ccc3n(S(=O)(=O)c3ccccc3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.37
CNR1 P21554 5/20 0.37
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
HSD17B10 Q99714 1/20 0.35
GAA P10253 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
APOBEC3A P31941 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726800 0.88 HTR6 (0.40) CNR2CNR1PSEN1PSEN2APH1B
SCHEMBL676120 0.83 HTR6 (0.44) ALDH1A1SMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL3730873 0.82 CNR2 (0.38) CNR2CNR1ALDH1A1SMN1; SMN2PSEN1
SCHEMBL676078 0.82 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2HPGDTSHRHSD17B10
SCHEMBL3669859 0.81 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2HPGDTSHRHSD17B10
SCHEMBL3721754 0.80 ALDH1A1 (0.40) CNR2ALDH1A1SMN1; SMN2PSEN1PSEN2
SCHEMBL3724854 0.80 PSEN1 (0.38) CNR2SMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL3724852 0.80 PSEN1 (0.38) CNR2SMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL3728544 0.79 NPC1 (0.42) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL3723156 0.77 NOD2 (0.37) ALDH1A1TSHRGAAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed