Picolamine

Picolamine

SCHEMBL3669942

COc1cc2nc(N3CCC(Cc4ccccc4)(C(=O)O)CC3)nc(O)c2cc1OC.NCc1cccnc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
WHR1 P49842 3/20 0.43
ADRA1A P35348 3/20 0.42
ADRA1B P35368 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Niacinamide SCHEMBL3669939 0.91 ADRA1A (0.44) WHR1ADRA1AADRA1B
SCHEMBL2170706 0.90 WHR1 (0.51) WHR1ADRA1AADRA1B
SCHEMBL2170268 0.87 PDGFRB (0.45) WHR1ADRA1AADRA1B
SCHEMBL13361589 0.85 WHR1 (0.49) WHR1ADRA1AADRA1B
SCHEMBL2188653 0.84 ADRA1A (0.49) ADRA1AADRA1B
SCHEMBL14715341 0.83 WHR1 (0.43) WHR1ADRA1AADRA1B
SCHEMBL2173344 0.82 ADRA1A (0.61) ADRA1AADRA1B
SCHEMBL2170928 0.81 L3MBTL1 (0.52)
SCHEMBL14715427 0.81 PDGFRB (0.43) WHR1ADRA1AADRA1B
SCHEMBL2170380 0.80 WHR1 (0.47) WHR1ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010054968-A1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-05-20 WO claimed