SCHEMBL3670130

SCHEMBL3670130

Cc1cc(OC2CCN(C(=O)O)CC2)ccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.48
GPR119 Q8TDV5 1/20 0.45
FFAR4 Q5NUL3 1/20 0.44
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
ACACB O00763 2/20 0.43
HRH3 Q9Y5N1 3/20 0.43
MRGPRX4 Q96LA9 1/20 0.42
PGR P06401 1/20 0.41
USP30 Q70CQ3 1/20 0.40
EPHX2 P34913 3/20 0.40
TBK1 Q9UHD2 1/20 0.40
FFAR1 O14842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3289631 0.85 PGR (0.55) ARPGREPHX2
SCHEMBL951252 0.85 GPR119 (0.65) ARGPR119HRH3
SCHEMBL216865 0.81 CCR5 (0.44) ACACBHRH3EPHX2
SCHEMBL21722970 0.80 BCL2A1 (0.44) ARGPR119FFAR4ACACBHRH3
SCHEMBL16483388 0.80 AR (0.48) ARFFAR4ACACBHRH3MRGPRX4
SCHEMBL16927539 0.79 FFAR4 (0.42) ARGPR119FFAR4PIK3CDPIK3CA
SCHEMBL16927540 0.79 FFAR4 (0.42) ARGPR119FFAR4PIK3CDPIK3CA
SCHEMBL26821604 0.79 AR (0.52) ARGPR119FFAR4PIK3CDPIK3CA
SCHEMBL2474849 0.79 USP30 (0.54) USP30
SCHEMBL3290157 0.79 HRH3 (0.64) GPR119HRH3EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2240441-A1 PROCESS FOR THE PREPARATION OF 6-SUBSTITUTED-1-(2H)-ISOQUINOLINONES Sanofi-Aventis (FR) 2010-10-20 EP disclosed
WO-2009080335-A1 PROCESS FOR THE PREPARATION OF 6-SUBSTITUTED-1-(2H)-ISOQUINOLINONES SANOFI-AVENTIS (FR) 2009-07-02 WO disclosed