SCHEMBL3671778

SCHEMBL3671778

O=C(c1cccc(Cl)c1)C1CNCCN1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
KDM2B Q8NHM5 4/20 0.43
SLC6A4 P31645 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
ADRB1 P08588 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41
HTT P42858 1/20 0.41
HTR3A P46098 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3801432 0.85 SIGMAR1 (0.46) HTR2CSIGMAR1
SCHEMBL3666620 0.85 SMN1; SMN2 (0.42) CYP2C9CYP2C19HTTMGLLSLC6A2
SCHEMBL5313826 0.77 HPGD (0.41) KDM2BSIGMAR1MGLL
SCHEMBL5263119 0.76 P4HB (0.38) HTR2CSIGMAR1
SCHEMBL11590269 0.75 SIGMAR1 (0.53) SIGMAR1
SCHEMBL8498078 0.74 SIGMAR1 (0.44) HTR2CSIGMAR1
SCHEMBL27523649 0.73 HTR2A (0.53) SLC6A4HTR3EHTR3BTP53CYP1A2
SCHEMBL3663206 0.72 DPP4 (0.43)
SCHEMBL3314213 0.71 HTR2C (0.44) NPSR1TP53HTR2AHTR2CHTR2B
SCHEMBL28214604 0.71 SIGMAR1 (0.41) HTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150532-A1 PIPERAZINE COMPOUNDS FOR THE INHIBITION OF HAEMATOPOIETIC PROSTAGLANDIN D SYNTHASE Evotec AG (DE) 2010-02-10 EP claimed
WO-2008122787-A1 PIPERAZINE COMPOUNDS FOR THE INHIBITION OF HAEMATOPOIETIC PROSTAGLANDIN D SYNTHASE EVOTEC AG (DE) 2008-10-16 WO claimed