SCHEMBL3672940

SCHEMBL3672940

NC1Oc2cccc(-c3cnc(C4CC4)nc3)c2C[C@@H]1N

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3672812 0.84 KCNH2 (0.38) DPP4
SCHEMBL3668903 0.81 SCN9A (0.41) DHFRDPP4
SCHEMBL3673795 0.81 DHFR (0.33) DHFRDPP4
SCHEMBL840895 0.81 SCN9A (0.36) DHFR
Ammonia Solution, Strong SCHEMBL3672937 0.80 SCN9A (0.35) DHFR
SCHEMBL3672628 0.76 SCN9A (0.41)
SCHEMBL3667284 0.73 KCNH2 (0.46) DPP4
SCHEMBL3670227 0.71 JAK3 (0.33) DPP4
SCHEMBL3674446 0.71 IDO1 (0.38)
SCHEMBL3730969 0.70 CREBBP (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2158198-A2 NOVEL N- (8HETEROARYLTETRAHYDRONAPHTALENE-2YL) OR N- (5- HETEROARYLCHROMANE-3-YL) CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN AstraZeneca AB (SE) 2010-03-03 EP disclosed
WO-2008130320-A2 NOVEL N- (8-HETEROARYLTETRAHYDRONAPHTALENE-2YL) OR N- (5- HETEROARYLCHROMANE-3-YL) CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed