SCHEMBL3673795

SCHEMBL3673795

CCc1ncc(-c2cccc3c2C[C@H](N)C(N)O3)cn1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.33
KCNH2 Q12809 2/20 0.31
SCN5A Q14524 2/20 0.31
SCN9A Q15858 2/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3672812 0.86 KCNH2 (0.38) KCNH2SCN5ASCN9ADPP4
SCHEMBL3668903 0.82 SCN9A (0.41) DHFRKCNH2SCN5ASCN9ADPP4
SCHEMBL3672940 0.81 DHFR (0.33) DHFRDPP4
SCHEMBL840902 0.80 SCN9A (0.38) DHFRKCNH2SCN5ASCN9A
Ammonia Solution, Strong SCHEMBL3673794 0.79 SCN9A (0.38) DHFRKCNH2SCN5ASCN9A
SCHEMBL3676949 0.76 SCN9A (0.38) KCNH2SCN5ASCN9ADPP4
SCHEMBL3672628 0.75 SCN9A (0.41) KCNH2SCN5ASCN9A
SCHEMBL3667284 0.75 KCNH2 (0.46) KCNH2SCN5ASCN9ADPP4
SCHEMBL3670227 0.72 JAK3 (0.33) DPP4
SCHEMBL3674498 0.72 DPP4 (0.40) DHFRDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2158198-A2 NOVEL N- (8HETEROARYLTETRAHYDRONAPHTALENE-2YL) OR N- (5- HETEROARYLCHROMANE-3-YL) CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN AstraZeneca AB (SE) 2010-03-03 EP disclosed
WO-2008130320-A2 NOVEL N- (8-HETEROARYLTETRAHYDRONAPHTALENE-2YL) OR N- (5- HETEROARYLCHROMANE-3-YL) CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed