SCHEMBL3672987

SCHEMBL3672987

O=Nc1c[nH]c(-c2ccccc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
MAPT P10636 4/20 0.44
KDM4E B2RXH2 3/20 0.44
CASP6 P55212 1/20 0.44
CYP1A2 P05177 3/20 0.41
PIN1 Q13526 2/20 0.41
CYP2C19 P33261 2/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
MTOR P42345 1/20 0.39
ADK P55263 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
DCUN1D1 Q96GG9 2/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
BTK Q06187 1/20 0.38
TNKS O95271 1/20 0.38
PARP1 P09874 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3933282 0.79 HPGDS (0.37) MEN1KMT2AMAPTKDM4ECASP6
SCHEMBL528246 0.72 MEN1 (0.46) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL27840974 0.71 MTOR (0.42) MEN1KMT2AKDM4ECYP1A2CYP2C19
SCHEMBL2094094 0.71 MTOR (0.42) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL27456927 0.71 MTOR (0.42) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL1954237 0.71 MTOR (0.42) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL637805 0.71 ALDH1A1 (0.48) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL3122569 0.71 MTOR (0.42) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL57159 0.71 NR1H2 (0.45) MEN1KMT2AMAPTKDM4ECYP1A2
SCHEMBL49612 0.71 GAA (0.52) MEN1KMT2AMAPTKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244460-B8 USE OF DIPYRIDINIUM COMPOUNDS FOR TREATING A DISEASE CHARACTERIZED BY PROLIFERATING CELLS CONTAINING NITRIC OXIDE SYNTHASE UNIV DUKE (US) 2010-05-19 EP disclosed
EP-1244460-A4 TREATMENTS BASED ON DISCOVERY THAT NITRIC OXIDE SYNTHASE IS A PARAQUAT DIAPHORASE UNIV DUKE (US) 2004-10-06 EP disclosed
EP-1244460-A1 TREATMENTS BASED ON DISCOVERY THAT NITRIC OXIDE SYNTHASE IS A PARAQUAT DIAPHORASE DUKE UNIVERSITY (US) 2002-10-02 EP disclosed
WO-2001028568-A1 TREATMENTS BASED ON DISCOVERY THAT NITRIC OXIDE SYNTHASE IS A PARAQUAT DIAPHORASE DUKE UNIVERSITY (US) 2001-04-26 WO disclosed