SCHEMBL3674201

SCHEMBL3674201

COc1cccc(OC)c1-c1ccc2c(c1)C(C[AsH2])CC2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.38
SYK P43405 2/20 0.38
JAK2 O60674 1/20 0.38
LCK P06239 1/20 0.38
KDR P35968 1/20 0.38
GSK3B P49841 1/20 0.38
LRRK2 Q5S007 1/20 0.38
HTR1A P08908 2/20 0.37
HTR7 P34969 2/20 0.37
POLL Q9UGP5 1/20 0.37
NQO2 P16083 3/20 0.37
MTNR1B P49286 3/20 0.37
CYP19A1 P11511 1/20 0.36
BRD4 O60885 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
ABCB1 P08183 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3642761 0.87 ADRA2A (0.42) MTNR1ASYKHTR1ADRD2DRD3
SCHEMBL3642020 0.79 GRIA1 (0.44) HTR1A
SCHEMBL3674205 0.78 AR (0.39) SYKJAK2LCKKDRGSK3B
SCHEMBL3642763 0.77 PDPK1 (0.49) DRD2DRD3
SCHEMBL3643157 0.77 ACHE (0.45) HTR1AHTR7POLLDRD2DRD3
SCHEMBL3646099 0.74 HTR2C (0.46) HTR1AHTR7
SCHEMBL13959050 0.71 ACHE (0.43) DRD2DRD3
SCHEMBL3642023 0.70 GRIA1 (0.44) DRD2DRD3
SCHEMBL3644416 0.70 GRIA1 (0.44) HTR1ADRD2DRD3
SCHEMBL3645246 0.70 ADRA2A (0.46) HTR7BRD4DRD2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173712-A2 INDANE-AMINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-04-14 EP claimed
WO-2009003719-A2 INDANE-AMINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2009-01-08 WO claimed