SCHEMBL3674766

SCHEMBL3674766

CCCNC(=O)c1ccc(-c2cnno2)cc1-c1cnno1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.46
RAB9A P51151 8/20 0.46
TP53 P04637 4/20 0.46
SMN1; SMN2 Q16637 5/20 0.45
POLB P06746 3/20 0.43
THRB P10828 1/20 0.43
RECQL P46063 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HPGD P15428 4/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
GAA P10253 1/20 0.40
KCNA3 P22001 3/20 0.39
CNR1 P21554 1/20 0.39
HTT P42858 1/20 0.39
HIF1A Q16665 1/20 0.39
KMT2A Q03164 2/20 0.37
HSD17B10 Q99714 1/20 0.37
CDK1 P06493 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551862 0.84 ROCK2 (0.38) NPC1RAB9AGAAGSK3B
SCHEMBL3674767 0.83 MAPK1 (0.48) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL4551736 0.78 ALDH1A1 (0.37) NPC1RAB9AALDH1A1GAAKMT2A
SCHEMBL30211623 0.66 POLB (0.61) SMN1; SMN2POLBTHRBRECQLTDP1
SCHEMBL22505247 0.66 POLB (0.61) SMN1; SMN2POLBTHRBRECQLTDP1
SCHEMBL11994154 0.64 CHRNB2 (0.64) SMN1; SMN2ALDH1A1LMNAGAAHTT
SCHEMBL17117168 0.62 NPC1 (1.00) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL26409544 0.62 POLB (0.56) SMN1; SMN2POLBTHRBRECQLTDP1
SCHEMBL9592081 0.61 POLB (0.55) NPC1RAB9ASMN1; SMN2POLBTHRB
SCHEMBL12349834 0.61 TP53 (0.78) NPC1RAB9ATP53SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2162136-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2010-03-17 EP disclosed
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed