SCHEMBL3677633

SCHEMBL3677633

C=CCc1ccc(-c2ccc(C(=O)O)cc2)cc1-c1ccc2c(c1)C(C)(C)CCC2(C)C

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARB P10826 16/20 0.76
RARG P13631 16/20 0.76
RARA P10276 14/20 0.76
RXRA P19793 6/20 0.66
RXRB P28702 3/20 0.51
RXRG P48443 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL498220 0.86 RARG (0.57) RARBRARGRARARXRA
SCHEMBL10040623 0.84 RARG (0.53) RARBRARGRARARXRA
SCHEMBL497953 0.82 RARB (0.87) RARBRARGRARARXRARXRB
SCHEMBL498280 0.81 RARB (0.76) RARBRARGRARARXRA
SCHEMBL5846340 0.80 RARB (0.77) RARBRARGRARARXRARXRB
SCHEMBL3677978 0.80 RARB (1.00) RARBRARGRARARXRARXRB
SCHEMBL7873016 0.78 RARB (0.83) RARBRARGRARARXRARXRB
SCHEMBL5846429 0.78 RARB (0.83) RARBRARGRARARXRARXRB
SCHEMBL5846624 0.78 RARB (0.83) RARBRARGRARARXRARXRB
SCHEMBL5846100 0.77 RARG (1.00) RARBRARGRARARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963249-B1 BIPHENYL DERIVATIVES AS SELECTIVE AGONISTS OF GAMMA RAR RECEPTORS GALDERMA RES & DEV (FR) 2010-07-28 EP disclosed
EP-1963249-B1 BIPHENYL DERIVATIVES AS SELECTIVE AGONISTS OF GAMMA RAR RECEPTORS GALDERMA RES & DEV (FR) 2010-07-28 EP disclosed
EP-1963249-A1 BIPHENYL DERIVATIVES AS SELECTIVE AGONISTS OF GAMMA RAR RECEPTORS Galderma Research & Development (FR) 2008-09-03 EP disclosed
WO-2007068579-A1 BIPHENYL DERIVATIVES AS SELECTIVE AGONISTS OF GAMMA RAR RECEPTORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2007-06-21 WO disclosed