SCHEMBL3680918

SCHEMBL3680918

CC1=C(C(=O)OS(=O)(=O)c2ccccc2)[C@@H](c2ccccc2Cl)C(C(=O)O)=C(COCCN)N1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.66
NR1I2 O75469 2/20 0.66
TBXA2R P21731 3/20 0.64
ADRA1A P35348 3/20 0.64
SLC6A3 Q01959 3/20 0.64
HTR1A P08908 2/20 0.64
ADRA2A P08913 2/20 0.64
CHRM1 P11229 2/20 0.64
DRD1 P21728 2/20 0.64
SLC6A2 P23975 2/20 0.64
OPRM1 P35372 2/20 0.64
DRD3 P35462 2/20 0.64
KCNH2 Q12809 2/20 0.64
ABCB11 O95342 2/20 0.64
ABCB1 P08183 2/20 0.64
ADORA3 P0DMS8 2/20 0.64
ADRB3 P13945 2/20 0.64
OPRK1 P41145 2/20 0.64
SCN5A Q14524 2/20 0.64
KCNK2 O95069 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2846050 1.00 CYP3A4 (0.66) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL3376883 0.93 CYP3A4 (0.77) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL34462108 0.88 TBXA2R (0.70) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL1610044 0.88 TBXA2R (0.70) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL16634960 0.88 TBXA2R (0.70) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
Benzene SCHEMBL7444141 0.88 TBXA2R (0.70) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL30669880 0.88 TBXA2R (0.70) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL2846047 0.88 CYP3A4 (0.75) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
SCHEMBL6299952 0.88 CYP3A4 (0.75) CYP3A4NR1I2TBXA2RADRA1ASLC6A3
Benzene SCHEMBL3268864 0.88 ABCB11 (0.82) CYP3A4NR1I2TBXA2RADRA1ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765342-B1 PHARMACEUTICAL COMPOSITION COMPRISING AMLODIPINE BESILATE AND LISINOPRIL DIHYDRATE AND PROCESS FOR THE PREPARATION THEREOF RICHTER GEDEON NYRT (HU) 2010-11-03 EP disclosed