SCHEMBL3685740

SCHEMBL3685740

CC(CN1CN(CC(C)N(C)C)CN(C[C@H](C)N(C)C)C1)N(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
ALOX15 P16050 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SLC22A1 O15245 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ESR1 P03372 1/20 0.34
PRNP P04156 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
HTR1A P08908 1/20 0.34
CHRM5 P08912 1/20 0.34
ADRA2A P08913 1/20 0.34
CALM1 P0DP23 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD2 P14416 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30364023 1.00 CYP2D6 (0.34) CYP2D6LMNACYP1A2ALOX15HSD17B10
SCHEMBL25838728 0.79 MEN1 (0.42) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL28638594 0.75 GAA (0.39) ALDH1A1HTR1AMC4RMAPTSMN1; SMN2
SCHEMBL8724143 0.74 CHRNB2 (0.34)
SCHEMBL3408660 0.74 SMN1; SMN2 (0.44) CYP2D6LMNACYP1A2ALOX15HSD17B10
SCHEMBL10867936 0.68 OPRK1 (0.44) CYP2D6OPRM1OPRK1
SCHEMBL1877599 0.65 TSHR (0.37) ALDH1A1DRD2DRD4PTGS1DRD3
SCHEMBL9761 0.63
SCHEMBL2268857 0.63
SCHEMBL28642676 0.62 GAA (0.37) ALDH1A1HTR1AMC4RSIGMAR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183232-A2 PI3 KINASE MODULATORS AND METHODS OF USE Amgen, Inc (US) 2010-05-12 EP claimed
WO-2009017822-A2 PI3 KINASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2009-02-05 WO claimed