SCHEMBL3685949

SCHEMBL3685949

COc1ccc(C(C)(C)C)cc1C=CC(=O)c1ccc(O)cc1N1CCN(C)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 3/20 0.47
NR1H4 Q96RI1 2/20 0.46
PTPN1 P18031 2/20 0.44
CHRNA7 P36544 2/20 0.44
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
BACE1 P56817 1/20 0.43
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAOB P27338 2/20 0.42
PARP1 P09874 1/20 0.42
MAOA P21397 1/20 0.42
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41
MAPK1 P28482 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686266 0.90 PDE4A (0.43) PTPN1PDE4APDE4BPDE4CPDE4D
SCHEMBL3685946 0.89 CHRNA7 (0.44) CAPN1NR1H4PTPN1CHRNA7BACE1
SCHEMBL3692417 0.89 CHRNA7 (0.44) CAPN1NR1H4PTPN1CHRNA7BACE1
SCHEMBL3687530 0.88 PTPN1 (0.55) PTPN1PDE4APDE4BPDE4CPDE4D
SCHEMBL3683957 0.85 CHRNA7 (0.40) CAPN1NR1H4PTPN1CHRNA7ALDH1A1
SCHEMBL3693475 0.80 SMN1; SMN2 (0.46) PTPN1PDE4BALDH1A1SMN1; SMN2MAOB
SCHEMBL3687529 0.80 SMN1; SMN2 (0.46) PTPN1PDE4BALDH1A1SMN1; SMN2MAOB
SCHEMBL3687761 0.79 HTR1A (0.44) PTPN1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL3686263 0.79 HTR1A (0.43) PTPN1ALDH1A1SMN1; SMN2MEN1MAPT
SCHEMBL3692486 0.79 HTR1A (0.43) PTPN1ALDH1A1SMN1; SMN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed