SCHEMBL3687761

SCHEMBL3687761

COc1ccc(C(C)(C)C)cc1C=CC(=O)c1c(F)cccc1N1CCN(C)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.44
HTR1D P28221 2/20 0.44
HTR1B P28222 2/20 0.44
HTR6 P50406 2/20 0.44
HTR2C P28335 1/20 0.44
KRAS P01116 1/20 0.43
TNFRSF1A P19438 2/20 0.43
ABCB1 P08183 2/20 0.42
ERAP1 Q9NZ08 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41
PTPN1 P18031 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3687530 0.85 PTPN1 (0.55) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3692364 0.81 HTR1A (0.44) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3687759 0.81 HTR1A (0.44) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3685949 0.79 CAPN1 (0.47) ABCB1SMN1; SMN2ALDH1A1PTPN1MEN1
SCHEMBL3686266 0.79 PDE4A (0.43) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3687529 0.79 SMN1; SMN2 (0.46) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3693475 0.79 SMN1; SMN2 (0.46) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3688318 0.79 NPY2R (0.46) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3686111 0.75 KRAS (0.47) HTR1AHTR1DHTR1BHTR6HTR2C
SCHEMBL3691974 0.75 RAB9A (0.51) SMN1; SMN2ALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed