SCHEMBL3685950

SCHEMBL3685950

Cc1ccccc1-c1ccc(N2CCN(C)CC2)cc1C=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
PKM P14618 1/20 0.48
ALDH1A1 P00352 4/20 0.48
HTR3A P46098 1/20 0.47
CSF1R P07333 1/20 0.45
PDK2 Q15119 1/20 0.44
CYP1A2 P05177 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAP4K1 Q92918 1/20 0.44
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
IDO2 Q6ZQW0 1/20 0.44
TACR1 P25103 1/20 0.44
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3685781 0.83 ADORA2A (0.51) NPC1RAB9APKMALDH1A1HTR3A
SCHEMBL5753256 0.77 MAPT (0.51) NPC1RAB9APKMALDH1A1HTR3A
SCHEMBL2913155 0.76 MAPT (0.56) NPC1RAB9AALDH1A1HTR3ACSF1R
SCHEMBL6868712 0.75 TACR1 (0.58) NPC1RAB9APKMALDH1A1HTR3A
SCHEMBL3696108 0.75 ALDH1A1 (0.50) ALDH1A1HTR3ACSF1RCYP1A2MEN1
SCHEMBL3688350 0.75 ALDH1A1 (0.52) NPC1RAB9APKMALDH1A1CYP1A2
SCHEMBL3685663 0.74 ALDH1A1 (0.56) NPC1RAB9APKMALDH1A1HTR3A
SCHEMBL3197069 0.74 MAPT (0.61) NPC1RAB9AALDH1A1HTR3AMEN1
SCHEMBL2908099 0.74 SIRT6 (0.60) ALDH1A1MAPK1
SCHEMBL2913153 0.74 TACR1 (0.57) ALDH1A1HTR3ACSF1RPDK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed