SCHEMBL3686478

SCHEMBL3686478

COc1cccc2c(CCC3(O)CCC(N)CC3)ccnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
PDE10A Q9Y233 1/20 0.36
ENPP1 P22413 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
PLAU P00749 1/20 0.34
MAPT P10636 5/20 0.34
TNF P01375 3/20 0.34
LITAF Q99732 3/20 0.34
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
ALOX12 P18054 3/20 0.34
HTT P42858 3/20 0.34
RAB9A P51151 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
NFKB1 P19838 1/20 0.34
MPI P34949 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3699154 0.79 HTR1A (0.36) HTR1AADRA1DADRA1AADRA1BMAPT
SCHEMBL3686475 0.76 KCNH2 (0.40) HTR1AADRA1DADRA1AADRA1BPDE10A
SCHEMBL3698422 0.74 KCNH2 (0.43)
SCHEMBL3698211 0.74 KCNA3 (0.36) HTR1AADRA1DADRA1AADRA1BMAPT
SCHEMBL16964453 0.73 HTR1A (0.60) HTR1AADRA1DADRA1AADRA1BPDE10A
SCHEMBL3687251 0.72 HTR1A (0.31) HTR1AADRA1DADRA1AADRA1B
SCHEMBL3688086 0.71 HTR1A (0.42) HTR1AADRA1DADRA1AADRA1BPDE10A
SCHEMBL3692453 0.71 HTR1A (0.49) HTR1AADRA1DADRA1AADRA1BENPP1
SCHEMBL16106422 0.70 HTR1A (0.54) HTR1AADRA1DADRA1AADRA1BPDE10A
SCHEMBL3694763 0.70 HTR1A (0.45) HTR1AADRA1DADRA1AADRA1BPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed