SCHEMBL3686475

SCHEMBL3686475

COc1cccc2c(CCC3(O)CCC(NCc4cc5ccccc5nc4Cl)CC3)ccnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.40
PDE10A Q9Y233 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
HTR1A P08908 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
TACR1 P25103 5/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
NFKB1 P19838 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686473 0.85 KCNH2 (0.49) KCNH2
SCHEMBL3688398 0.77 KCNH2 (0.52) KCNH2
SCHEMBL3699154 0.77 HTR1A (0.36) KCNH2ALDH1A1MAPTHTR1AADRA1D
SCHEMBL3686478 0.76 HTR1A (0.43) PDE10AALDH1A1MAPTHTR1AADRA1D
SCHEMBL3687251 0.71 HTR1A (0.31) KCNH2HTR1AADRA1DADRA1AADRA1B
SCHEMBL3686499 0.69 KCNH2 (0.50) KCNH2
SCHEMBL3689424 0.66 HTR1A (0.44) KCNH2ALDH1A1HTR1AADRA1DADRA1A
SCHEMBL5772791 0.65 KCNH2 (0.37) KCNH2ALDH1A1HTR1AADRA1DADRA1A
SCHEMBL3687247 0.64 KCNH2 (0.56) KCNH2
SCHEMBL13145887 0.64 KCNH2 (0.58) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed