SCHEMBL3687251

SCHEMBL3687251

COc1cccc2c(CCC3(O)CCC(NCC4=C(C5=COC(O)=CO5)CCC=C4)CC3)ccnc12

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
KCNH2 Q12809 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5649014 0.84 KCNH2 (0.42) KCNH2
SCHEMBL3688398 0.73 KCNH2 (0.52) KCNH2
SCHEMBL3686478 0.72 HTR1A (0.43) HTR1AADRA1DADRA1AADRA1B
SCHEMBL3686475 0.71 KCNH2 (0.40) HTR1AADRA1DADRA1AADRA1BKCNH2
SCHEMBL3699154 0.71 HTR1A (0.36) HTR1AADRA1DADRA1AADRA1BKCNH2
SCHEMBL3687395 0.70
SCHEMBL6219493 0.62 KCNH2 (0.45) HTR1AADRA1DADRA1AADRA1BKCNH2
SCHEMBL3698211 0.61 KCNA3 (0.36) HTR1AADRA1DADRA1AADRA1B
SCHEMBL3688086 0.61 HTR1A (0.42) HTR1AADRA1DADRA1AADRA1BKCNH2
SCHEMBL3689424 0.61 HTR1A (0.44) HTR1AADRA1DADRA1AADRA1BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed