SCHEMBL3686783

SCHEMBL3686783

COc1ccc(C(C)(C)C#N)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.39
HTR2A P28223 2/20 0.39
KCNH2 Q12809 1/20 0.36
NQO1 P15559 1/20 0.36
KDM4E B2RXH2 3/20 0.36
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
GFER P55789 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17162836 0.86 MAPT (0.36) SLC6A4HTR2AKCNH2NQO1KDM4E
SCHEMBL11708277 0.81 CA12 (0.48) KDM4EARALDH1A1MAPTMEN1
SCHEMBL8225342 0.80 CA1 (0.45) SLC6A4HTR2AKCNH2KDM4ESLC6A2
SCHEMBL3993767 0.79 KIF11 (0.43) NQO1KDM4EPGRARALDH1A1
SCHEMBL837308 0.78 TSHR (0.52) MEN1TSHRKMT2AHSD17B10
SCHEMBL11258529 0.77 ALDH1A1 (0.49) ARALDH1A1MAPTMEN1KMT2A
SCHEMBL7765888 0.76 NQO1 (0.36) NQO1KDM4EPGRARALDH1A1
SCHEMBL16518005 0.76 AR (0.39) NQO1KDM4EPGRARALDH1A1
SCHEMBL9458157 0.75 IDO1 (0.33) TSHR
SCHEMBL307319 0.75 PYCR1 (0.34) SLC6A4HTR2AKCNH2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
US-20060052600-A1 Amino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-03-09 US disclosed
EP-1506157-A2 AMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed
WO-2003097575-A2 AMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed