SCHEMBL3689424

SCHEMBL3689424

COc1cccc2c(CNC3CCCNCC3)ccnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TACR1 P25103 4/20 0.40
KCNH2 Q12809 2/20 0.39
ALDH1A1 P00352 2/20 0.39
JUND P17535 1/20 0.39
FOSB P53539 1/20 0.39
USP2 O75604 1/20 0.38
CYP2D6 P10635 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218091 0.82 HTR1A (0.45) HTR1AADRA1DADRA1AADRA1BCYP1A2
SCHEMBL3689420 0.77 KCNH2 (0.52) KDM4EGAAHTTKCNH2ALDH1A1
SCHEMBL3692137 0.75 MEN1 (0.49) MEN1KMT2A
SCHEMBL8821601 0.74 KDM1A (0.56) MEN1KMT2AKDM4EGAAHTT
SCHEMBL8821304 0.74 TACR1 (0.50) TACR1
SCHEMBL8696023 0.74 MEN1 (0.60) MEN1KMT2AGAATACR1ALDH1A1
SCHEMBL29862532 0.72 HTR1A (0.55) HTR1AADRA1DADRA1AADRA1BCYP1A2
SCHEMBL24716111 0.72 HTR2C (0.56) HTR1AADRA1DADRA1AADRA1BJUND
SCHEMBL30626631 0.72 HTR2C (0.56) HTR1AADRA1DADRA1AADRA1BJUND
Hydrochloric Acid SCHEMBL23360306 0.71 HTR1A (0.54) HTR1AADRA1DADRA1AADRA1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed