SCHEMBL3692137

SCHEMBL3692137

COc1cccc2c(CNC3CCCN(CCCc4ccccc4)CC3)ccnc12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
POLB P06746 1/20 0.49
KMT2A Q03164 1/20 0.49
BCHE P06276 3/20 0.48
ACHE P22303 3/20 0.48
BACE1 P56817 3/20 0.48
SIGMAR1 Q99720 1/20 0.45
GRIN2B Q13224 1/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD4 P21917 1/20 0.41
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692134 0.82 KCNH2 (0.61) MEN1KMT2A
SCHEMBL13145572 0.77 KCNH2 (0.65)
SCHEMBL3689424 0.75 HTR1A (0.44) MEN1KMT2A
SCHEMBL9753832 0.73 MEN1 (0.57) MEN1POLBKMT2ABCHEACHE
SCHEMBL6628061 0.70 HTR1A (0.54) MEN1KMT2ABCHEACHESIGMAR1
SCHEMBL16964628 0.70 BCHE (0.55) MEN1KMT2ABCHE
SCHEMBL6975733 0.69 HTR4 (0.48) BCHEACHESIGMAR1
SCHEMBL5754351 0.69 SIGMAR1 (0.47) SIGMAR1
SCHEMBL5760090 0.69 ABCB1 (0.47) SIGMAR1ABCB1
SCHEMBL14514811 0.68 KCNH2 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed