SCHEMBL3690486

SCHEMBL3690486

CN(Cc1cc(-c2cccnc2F)c(S(=O)(=O)c2ncc[nH]2)s1)C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.34
CACNA1G O43497 1/20 0.32
CACNA1B Q00975 1/20 0.32
CACNA1C Q13936 1/20 0.32
AGTR2 P50052 2/20 0.31
SSTR4 P31391 1/20 0.31
GLS O94925 1/20 0.31
HTR2C P28335 2/20 0.31
SLC6A4 P31645 2/20 0.31
SOS1 Q07889 1/20 0.31
HTR2A P28223 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3703108 0.94 PDK2 (0.31) PDK2AGTR2GLSSOS1
SCHEMBL4125938 0.88 FFAR4 (0.34) FFAR4
SCHEMBL3649951 0.86 PDK2 (0.35) PDK2CACNA1GCACNA1BCACNA1CGLS
SCHEMBL3654948 0.86 F2 (0.35) PDK2AGTR2GLSHTR2CSLC6A4
SCHEMBL3804721 0.84 ABCC9 (0.33) PDK2CACNA1GCACNA1BCACNA1CGLS
SCHEMBL3652358 0.84 GLS (0.32) PDK2GLSHTR2CSLC6A4SOS1
SCHEMBL4530415 0.84 PDK2 (0.32) PDK2SSTR4GLSHTR2CSLC6A4
SCHEMBL3651630 0.83 HTR2C (0.32) PDK2AGTR2SSTR4GLSHTR2C
SCHEMBL3690491 0.83 FFAR4 (0.32) FFAR4
SCHEMBL3803075 0.82 ALDH1A1 (0.33) PDK2AGTR2HTR2CSLC6A4SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed