SCHEMBL369177

SCHEMBL369177

Cc1cc(Cl)ccc1C(CC(=NO)C1=CC=CN(C)C1)c1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.33
CA2 P00918 11/20 0.32
CA1 P00915 10/20 0.32
CA9 Q16790 9/20 0.32
CA12 O43570 8/20 0.32
CHRNA7 P36544 2/20 0.31
CA4 P22748 2/20 0.31
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
CA7 P43166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370503 0.84 GPBAR1 (0.46) GPBAR1KEAP1NFE2L2
SCHEMBL369976 0.82 GPBAR1 (0.35) GPBAR1
SCHEMBL370694 0.80 GPBAR1 (0.37) GPBAR1KEAP1NFE2L2
SCHEMBL369724 0.77 GPBAR1 (0.38) GPBAR1CA2CA1CA9CA12
SCHEMBL369725 0.77 GPBAR1 (0.38) GPBAR1CA2CA1CA9CA12
SCHEMBL369726 0.77 GPBAR1 (0.38) GPBAR1CA2CA1CA9CA12
SCHEMBL10241381 0.75 GPBAR1 (0.40) GPBAR1CA2CA1CA9CA12
SCHEMBL10241383 0.75 GPBAR1 (0.40) GPBAR1CA2CA1CA9CA12
SCHEMBL1390699 0.75 GPBAR1 (0.40) GPBAR1CA2CA1CA9CA12
SCHEMBL370177 0.75 GPBAR1 (0.40) GPBAR1CA2CA1CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed