SCHEMBL369976

SCHEMBL369976

Cc1cc(Cl)ccc1C(CC(=NO)C1=CC=CN(C)C1)c1ccc(C(=O)NCCS(C)(=O)=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.35
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33
MDM2 Q00987 1/20 0.33
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
GCGR P47871 2/20 0.31
EPHX2 P34913 3/20 0.31
GCG P01275 1/20 0.31
CYP11B2 P19099 1/20 0.30
TMEM97 Q5BJF2 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370694 0.86 GPBAR1 (0.37) GPBAR1ALDH1A1GCGRGCG
SCHEMBL370503 0.83 GPBAR1 (0.46) GPBAR1
SCHEMBL369177 0.82 GPBAR1 (0.33) GPBAR1
SCHEMBL369287 0.82 GPBAR1 (0.36) GPBAR1LMNATP53MDM2ALDH1A1
SCHEMBL369285 0.82 GPBAR1 (0.36) GPBAR1LMNATP53MDM2ALDH1A1
SCHEMBL369286 0.82 GPBAR1 (0.36) GPBAR1LMNATP53MDM2ALDH1A1
SCHEMBL363112 0.79 GPBAR1 (0.36) GPBAR1TP53MDM2ALDH1A1POLB
SCHEMBL1390151 0.75 EPHX2 (0.35) GPBAR1LMNATP53MDM2GCGR
SCHEMBL1390150 0.75 EPHX2 (0.35) GPBAR1LMNATP53MDM2GCGR
SCHEMBL368212 0.75 TP53 (0.36) LMNATP53MDM2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed